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Home/Compounds/CAS 162401-32-3
Formula C17H14Cl2F2N2O3MW 403.2Research-use catalog entryCOA/SDS by request

Roflumilast

CAS Number: 162401-32-3

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99%
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Loading RDKit molecule structure...
InChIKey: MNDBXUUTURYVHR-UHFFFAOYSA-NC17H14Cl2F2N2O3 | MW 403.2

Chemical Absolute Identifiers

CAS Number

162401-32-3

PubChem CID

449193

Molecular Formula

C17H14Cl2F2N2O3

Molecular Weight

403.2 g/mol

Exact Mass

402.034954

InChIKey

MNDBXUUTURYVHR-UHFFFAOYSA-N

IUPAC Name

3-(cyclopropylmethoxy)-N-(3,5-dichloro-4-pyridinyl)-4-(difluoromethoxy)benzamide

SMILES String

C1CC1COC2=C(C=CC(=C2)C(=O)NC3=C(C=NC=C3Cl)Cl)OC(F)F

Physical Properties

pKa

8.74

Properties are provided as catalog reference data and may be confirmed through supplier documentation when required.

Catalog Facts

Structural features

Roflumilast (CAS 162401-32-3) is listed in the Pharmaceutical Intermediates portfolio, with molecular formula C17H14Cl2F2N2O3 and molecular weight 403. 20 g/mol.

Sourcing context

Catalog reference for RFQ preparation, supplier confirmation, and research chemical sourcing review.

Research use context

Intended for research-stage medicinal chemistry and intermediate synthesis workflows; structure-derived tags include nitrogen-containing heterocycle.

Documentation needs

COA/SDS status, availability, lead time, pack size, and shipment documentation can be confirmed during quotation.

Applications & Classification

Pharmaceutical Intermediate ResearchResearch intermediateCustom synthesis building blockPharmaceutical intermediate researchResearch chemical sourcingCustom synthesis and catalog availability reviewCOA, SDS, pricing, and fulfillment workflow
Biological target reference

ChEMBL reports experimental activity evidence for: 3',5'-cyclic-AMP phosphodiesterase 4D (Homo sapiens) — 26 assays; 3',5'-cyclic-AMP phosphodiesterase 4B (Homo sapiens) — 34 assays; 3',5'-cyclic-AMP phosphodiesterase 4A (Homo sapiens) — 4 assays; 3',5'-cyclic-AMP phosphodiesterase 4C (Homo sapiens) — 2 assays; Histone-lysine N-methyltransferase SETD7 (Homo sapiens) — 3 assays. These records describe research assays and do not establish therapeutic efficacy or clinical use.

3',5'-cyclic-AMP phosphodiesterase 4D

Homo sapiens · SINGLE PROTEIN · 26 qualifying assays · 26 documents · best pChEMBL 9.89

Experimental evidence source: ChEMBL

3',5'-cyclic-AMP phosphodiesterase 4B

Homo sapiens · SINGLE PROTEIN · 34 qualifying assays · 30 documents · best pChEMBL 9.82

Experimental evidence source: ChEMBL

3',5'-cyclic-AMP phosphodiesterase 4A

Homo sapiens · SINGLE PROTEIN · 4 qualifying assays · 4 documents · best pChEMBL 9.68

Experimental evidence source: ChEMBL

3',5'-cyclic-AMP phosphodiesterase 4C

Homo sapiens · SINGLE PROTEIN · 2 qualifying assays · 2 documents · best pChEMBL 8.77

Experimental evidence source: ChEMBL

Histone-lysine N-methyltransferase SETD7

Homo sapiens · SINGLE PROTEIN · 3 qualifying assays · 1 documents

Experimental evidence source: ChEMBL

Safety & Handling

Safety and handling reference content is available through documentation requests.

For supplier-issued SDS, request documentation before handling, storage, shipment, or procurement decisions.

Preliminary Safety Reference

For supplier-issued SDS or COA, submit a documentation request.

Safety Reference / SDS Request

Names & Synonyms / External Identifiers

Chemical Name

Roflumilast

Names & Synonyms

DAXAS3-(CYCLOPROPYLMETHOXY)-N-(3,5-DICHLOROPYRIDIN-4-YL)-4-(DIFLUOROMETHOXY)BENZAMIDEDalirespBY217Benzamide, 3-(cyclopropylmethoxy)-N-(3,5-dichloro-4-pyridinyl)-4-(difluoromethoxy)-
Show all synonyms
ZORYVEroflumilastumARQ-154 (Roflumilast foam)3-cyclopropylmethoxy-4-difluoromethoxy-N-(3,5-di-chloropyrid-4-yl)benzamide3-Cyclopropylmethoxy-N-(3,5-dichloropyridin-4-yl)-4-(difluoromethoxy)benzamideC17H14Cl2F2N2O3BY 217Roflumilast (Daxas)B 9302-107ROFLibertekRoflumilast [USAN]Roflumilast [USAN:INN]Roflumilast (JAN/USAN/INN)
External Identifiers
EC NUMBER: 685-382-2DSSTOX SUBSTANCE ID: DTXSID8044123CHEMBL ID: CHEMBL193240CHEBI ID: CHEBI:47657UNII: 0P6C6ZOP5UDRUGBANK ID: DB01656HMDB ID: HMDB0257288KEGG ID: D05744METABOLOMICS WORKBENCH ID: 56780NCI THESAURUS CODE: C76890PHARMGKB ID: PA165948052RXCUI: 1091836WIKIDATA ID: Q693482
Literature & Patent References
DOI 10.1016/j.bmc.2025.118067An overview of small-molecule agents for the treatment of psoriasis.DOI 10.1021/acs.jmedchem.4c02969Design, Synthesis, and Evaluation of Selective PDE4 Inhibitors for the Therapy of Pulmonary Injury.DOI 10.1021/acs.jmedchem.5c00266Structure-Based Optimization of Moracin M as Potent and Selective PDE4 Inhibitors with Antipsoriasis Effects.DOI 10.1021/acs.jmedchem.5c00505Design, Synthesis, and Biological Evaluation of New PDE4 Inhibitors for the Treatment of Pressure Ulcers.PMID 39832444An overview of small-molecule agents for the treatment of psoriasis.PMID 39847693Design, Synthesis, and Evaluation of Selective PDE4 Inhibitors for the Therapy of Pulmonary Injury.PMID 40066994Structure-Based Optimization of Moracin M as Potent and Selective PDE4 Inhibitors with Antipsoriasis Effects.PMID 40423264Design, Synthesis, and Biological Evaluation of New PDE4 Inhibitors for the Treatment of Pressure Ulcers.

Documentation & Compliance Facts

Compliance Facts

Shipment review: Required

Documentation available by request

Certificate of Analysis (COA): By request

Supplier Safety Data Sheet (SDS): By request

Purity and pack size confirmation: By request

Availability and lead time review: Confirmed by RFQ

Shipment documentation review: By request

For supplier-issued documentation by request, use the RFQ actions on this page.Review preliminary safety reference

What happens after RFQ

  1. 1We review the CAS identity, quantity, and documentation request.
  2. 2We check sourcing options, supplier availability, COA/SDS, purity, pack size, and lead time.
  3. 3We review destination and shipment documentation needs when applicable.
  4. 4We follow up with a quotation or clarification request.

Text Reference Cues

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Non-public related references

3-(Cyclopropylmethoxy)-4-(difluoromethoxy)benzoic AcidCAS 162401-62-9
3-(Cyclopropylmethoxy)-4-(difluoromethoxy)benzaldehydeCAS 151103-09-2
N-(3,5-dichloropyridin-4-yl)-3,4-dihydroxybenzamideCAS 1412448-29-3
Methyl 3-(cyclopropylmethoxy)-4-hydroxybenzoateCAS 848574-60-7
3-(Cyclopropylmethoxy)-4-hydroxybenzoic acidCAS 1243391-44-7

Non-public references are shown as text only and do not imply equivalence, availability, or shared use.

Catalog navigation

Related Catalog Entries

Other public CAS pages in this catalog. These links support navigation across additional intermediates and do not imply equivalence, availability, or shared use.

CAS 162401-62-93-(Cyclopropylmethoxy)-4-(difluoromethoxy)benzoic AcidCAS 151103-09-23-(Cyclopropylmethoxy)-4-(difluoromethoxy)benzaldehydeCAS 1412448-29-3N-(3,5-dichloropyridin-4-yl)-3,4-dihydroxybenzamideCAS 22994-85-0BenznidazoleCAS 114-07-8ErythromycinCAS 181695-72-7ValdecoxibCAS 608141-41-9ApremilastCAS 433695-36-4N,N,2-trimethyl-5-nitrobenzenesulfonamideCAS 1002310-00-0Tert-butyl 1-(2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)ethylcarbamateCAS 1005174-17-3(E)-3-(2-Propyl-6-(trifluoromethyl)pyridin-3-yl)acrylic acid

RFQ questions for CAS 162401-32-3

What are the key identifiers for Roflumilast (CAS 162401-32-3)?

Roflumilast is identified by CAS 162401-32-3, with molecular formula C17H14Cl2F2N2O3, molecular weight 403.2, InChIKey MNDBXUUTURYVHR-UHFFFAOYSA-N.

Does CAS 162401-32-3 have reported biological target evidence?

ChEMBL contains qualifying experimental assay evidence associated with 3',5'-cyclic-AMP phosphodiesterase 4D, 3',5'-cyclic-AMP phosphodiesterase 4B, 3',5'-cyclic-AMP phosphodiesterase 4A, 3',5'-cyclic-AMP phosphodiesterase 4C, Histone-lysine N-methyltransferase SETD7. These records do not establish therapeutic efficacy or clinical use.

Can I request a COA for CAS 162401-32-3?

Yes. Submit an RFQ and specify COA requirements. Lot-specific COA depends on supplier confirmation.

Can I request supplier SDS for Roflumilast?

Yes. Supplier SDS can be requested through the RFQ workflow before handling, storage, shipment, or procurement decisions.

Is CAS 162401-32-3 available for quotation?

Availability, pack size, lead time, and pricing are confirmed through RFQ.

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