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Home/Compounds/CAS 23491-48-7
Formula C11H16N4O2MW 236.27Research-use catalog entryCOA/SDS by request

5-(4-Methylpiperazin-1-yl)-2-nitroaniline

CAS Number: 23491-48-7

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Loading RDKit molecule structure...
InChIKey: MWLBMGPQZJDFKZ-UHFFFAOYSA-NC11H16N4O2 | MW 236.27

Chemical Absolute Identifiers

CAS Number

23491-48-7

PubChem CID

2760034

Molecular Formula

C11H16N4O2

Molecular Weight

236.27 g/mol

Exact Mass

236.127326

InChIKey

MWLBMGPQZJDFKZ-UHFFFAOYSA-N

SMILES String

CN1CCN(c2ccc([N+](=O)[O-])c(N)c2)CC1

Physical Properties

No physical property values available.

Properties are provided as catalog reference data and may be confirmed through supplier documentation when required.

Catalog Facts

Structural features

5-(4-Methylpiperazin-1-yl)-2-nitroaniline (CAS 23491-48-7) is listed in the Pharmaceutical Intermediates portfolio, with molecular formula C11H16N4O2 and molecular weight 236. 27 g/mol.

Sourcing context

Catalog reference for RFQ preparation, supplier confirmation, and research chemical sourcing review.

Research use context

Intended for research-stage medicinal chemistry and intermediate synthesis workflows; structure-derived tags include nitrogen-containing heterocycle.

Documentation needs

COA/SDS status, availability, lead time, pack size, and shipment documentation can be confirmed during quotation.

Applications & Classification

Pharmaceutical Intermediate ResearchResearch intermediateCustom synthesis building blockPharmaceutical intermediate researchResearch chemical sourcingCustom synthesis and catalog availability reviewCOA, SDS, pricing, and fulfillment workflow
Biological target reference

ChEMBL reports experimental activity evidence for: NAD-dependent protein deacylase sirtuin-6 (Homo sapiens) — 5 assays; Geminin (Homo sapiens) — 2 assays. These records describe research assays and do not establish therapeutic efficacy or clinical use.

NAD-dependent protein deacylase sirtuin-6

Homo sapiens · SINGLE PROTEIN · 5 qualifying assays · 1 documents · best pChEMBL 5.31

Experimental evidence source: ChEMBL

Geminin

Homo sapiens · SINGLE PROTEIN · 2 qualifying assays · 1 documents

Experimental evidence source: ChEMBL

Safety & Handling

Safety and handling reference content is available through documentation requests.

For supplier-issued SDS, request documentation before handling, storage, shipment, or procurement decisions.

Preliminary Safety Reference

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Safety Reference / SDS Request

Names & Synonyms / External Identifiers

Chemical Name

5-(4-Methylpiperazin-1-yl)-2-nitroaniline

Names & Synonyms

5-(4-Methylpiperazin-1-yl)-2-nitrophenylamine5-(4-methylpiperazino)-2-nitroaniline5-(4-Methyl-piperazin-1-yl)-2-nitro-phenylamine5-(4-methylpiperazin-1-yl)-2-nitrobenzenamine5-(4-Methyl-piperazin-1-yl)-2-nitroaniline
Show all synonyms
5-(4-methylpiperazinyl)-2-nitrophenylamine5-(4-Methyl-1-piperazinyl)-2-nitroaniline5-(4-methylpiperazin-1-yl)-2-nitro-aniline1-{3-amino-4-nitrophenyl}-4-methylpiperazineOprea1_384504benzenamine, 5-(4-methyl-1-piperazinyl)-2-nitro-AG-690/33045044
External Identifiers
EC NUMBER: 673-328-0DSSTOX SUBSTANCE ID: DTXSID20374997CHEMBL ID: CHEMBL1370863WIKIDATA ID: Q72495674
Experimental Spectrum References
13C NMR SpectraVapor Phase IR Spectra
Literature & Patent References
DOI 10.1021/acs.jmedchem.4c01223Discovery of Novel PROTAC SIRT6 Degraders with Potent Efficacy against Hepatocellular Carcinoma.PMID 39323022Discovery of Novel PROTAC SIRT6 Degraders with Potent Efficacy against Hepatocellular Carcinoma.DOI 10.1016/j.bmcl.2020.127215Discovery of 5-(4-methylpiperazin-1-yl)-2-nitroaniline derivatives as a new class of SIRT6 inhibitors.PMID 32631504Discovery of 5-(4-methylpiperazin-1-yl)-2-nitroaniline derivatives as a new class of SIRT6 inhibitors.

Documentation & Compliance Facts

Compliance Facts

Shipment review: Required

Documentation available by request

Certificate of Analysis (COA): By request

Supplier Safety Data Sheet (SDS): By request

Purity and pack size confirmation: By request

Availability and lead time review: Confirmed by RFQ

Shipment documentation review: By request

For supplier-issued documentation by request, use the RFQ actions on this page.Review preliminary safety reference

What happens after RFQ

  1. 1We review the CAS identity, quantity, and documentation request.
  2. 2We check sourcing options, supplier availability, COA/SDS, purity, pack size, and lead time.
  3. 3We review destination and shipment documentation needs when applicable.
  4. 4We follow up with a quotation or clarification request.

Text Reference Cues

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Non-public related references

4-(4-Methylpiperazin-1-yl)benzoic acidCAS 86620-62-4
1-Ethyl-4-(4-nitrophenyl)piperazineCAS 115619-00-6
4-(4-(4-Methyl-1-piperazinyl)-1-piperidinyl)benzenamineCAS 959795-70-1
1-Methyl-4-(4-nitro-2-(trifluoromethyl)benzyl)piperazineCAS 694499-24-6
1-(6-Nitropyridin-3-yl)piperazineCAS 775288-71-6

Non-public references are shown as text only and do not imply equivalence, availability, or shared use.

Catalog navigation

Related Catalog Entries

Other public CAS pages in this catalog. These links support navigation across additional intermediates and do not imply equivalence, availability, or shared use.

CAS 86620-62-44-(4-Methylpiperazin-1-yl)benzoic acidCAS 115619-00-61-Ethyl-4-(4-nitrophenyl)piperazineCAS 109-01-31-MethylpiperazineCAS 1635-61-65-Chloro-2-nitroanilineCAS 182618-86-61-Boc-4-(4-Nitrophenyl)piperazineCAS 1002310-00-0Tert-butyl 1-(2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)ethylcarbamateCAS 1005174-17-3(E)-3-(2-Propyl-6-(trifluoromethyl)pyridin-3-yl)acrylic acidCAS 1018125-49-92-(3-Cyclopropyl-6-ethyl-4-(trifluoromethyl)-1H-pyrazolo[3,4-b]pyridin-1-yl)acetic acidCAS 1018128-07-8Isopropyl 4-chloro-2-methylquinoline-6-carboxylateCAS 1018142-22-76-cyclopropyl-1-(2,2-difluoroethyl)-3-methyl-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid

RFQ questions for CAS 23491-48-7

What are the key identifiers for 5-(4-Methylpiperazin-1-yl)-2-nitroaniline (CAS 23491-48-7)?

5-(4-Methylpiperazin-1-yl)-2-nitroaniline is identified by CAS 23491-48-7, with molecular formula C11H16N4O2, molecular weight 236.27, InChIKey MWLBMGPQZJDFKZ-UHFFFAOYSA-N.

Does CAS 23491-48-7 have reported biological target evidence?

ChEMBL contains qualifying experimental assay evidence associated with NAD-dependent protein deacylase sirtuin-6, Geminin. These records do not establish therapeutic efficacy or clinical use.

Can I request a COA for CAS 23491-48-7?

Yes. Submit an RFQ and specify COA requirements. Lot-specific COA depends on supplier confirmation.

Can I request supplier SDS for 5-(4-Methylpiperazin-1-yl)-2-nitroaniline?

Yes. Supplier SDS can be requested through the RFQ workflow before handling, storage, shipment, or procurement decisions.

Is CAS 23491-48-7 available for quotation?

Availability, pack size, lead time, and pricing are confirmed through RFQ.

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