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Home/Compounds/CAS 459789-99-2
Formula C26H44O4MW 420.6Research-use catalog entryCOA/SDS by request

Obeticholic Acid

CAS Number: 459789-99-2

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Loading RDKit molecule structure...
InChIKey: ZXERDUOLZKYMJM-ZWECCWDJSA-NC26H44O4 | MW 420.6

Chemical Absolute Identifiers

CAS Number

459789-99-2

PubChem CID

447715

Molecular Formula

C26H44O4

Molecular Weight

420.6 g/mol

Exact Mass

420.32396

InChIKey

ZXERDUOLZKYMJM-ZWECCWDJSA-N

IUPAC Name

(4R)-4-[(3R,5S,6R,7R,8S,9S,10S,13R,14S,17R)-6-ethyl-3,7-dihydroxy-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]pentanoic acid

SMILES String

CC[C@@H]1[C@@H]2C[C@@H](CC[C@@]2([C@H]3CC[C@]4([C@H]([C@@H]3[C@@H]1O)CC[C@@H]4[C@H](C)CCC(=O)O)C)C)O

Physical Properties

pKa

4.76

Properties are provided as catalog reference data and may be confirmed through supplier documentation when required.

Catalog Facts

Structural features

Obeticholic Acid (CAS 459789-99-2) is listed in the Pharmaceutical Intermediates portfolio, with molecular formula C26H44O4 and molecular weight 420. 60 g/mol.

Sourcing context

Catalog reference for RFQ preparation, supplier confirmation, and research chemical sourcing review.

Research use context

Intended for research-stage medicinal chemistry and intermediate synthesis workflows.

Documentation needs

COA/SDS status, availability, lead time, pack size, and shipment documentation can be confirmed during quotation.

Applications & Classification

Enzyme ResearchPharmaceutical Intermediate ResearchResearch intermediateCustom synthesis building blockPharmaceutical intermediate researchResearch chemical sourcingCustom synthesis and catalog availability reviewCOA, SDS, pricing, and fulfillment workflow
Biological target reference

ChEMBL reports experimental activity evidence for: Bile acid receptor (Homo sapiens) — 65 assays; G-protein coupled bile acid receptor 1 (Homo sapiens) — 16 assays; G-protein coupled bile acid receptor 1 (Mus musculus) — 2 assays; Alpha-1A adrenergic receptor (Homo sapiens) — 4 assays; Alpha-2A adrenergic receptor (Homo sapiens) — 3 assays. These records describe research assays and do not establish therapeutic efficacy or clinical use.

Bile acid receptor

Homo sapiens · SINGLE PROTEIN · 65 qualifying assays · 34 documents · best pChEMBL 8

Experimental evidence source: ChEMBL

G-protein coupled bile acid receptor 1

Homo sapiens · SINGLE PROTEIN · 16 qualifying assays · 10 documents · best pChEMBL 7.62

Experimental evidence source: ChEMBL

G-protein coupled bile acid receptor 1

Mus musculus · SINGLE PROTEIN · 2 qualifying assays · 1 documents · best pChEMBL 5.24

Experimental evidence source: ChEMBL

Alpha-1A adrenergic receptor

Homo sapiens · SINGLE PROTEIN · 4 qualifying assays · 1 documents · best pChEMBL 5.2

Experimental evidence source: ChEMBL

Alpha-2A adrenergic receptor

Homo sapiens · SINGLE PROTEIN · 3 qualifying assays · 1 documents · best pChEMBL 4.96

Experimental evidence source: ChEMBL

Safety & Handling

Safety and handling reference content is available through documentation requests.

For supplier-issued SDS, request documentation before handling, storage, shipment, or procurement decisions.

Preliminary Safety Reference

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Safety Reference / SDS Request

Names & Synonyms / External Identifiers

Chemical Name

Obeticholic Acid

Names & Synonyms

6-Ethylchenodeoxycholic acidOcaliva6-Ethyl-CDCAacido obeticolicoacide obeticholique
Show all synonyms
INT 7476alpha-ethylchenodeoxycholic acid6alpha-ethyl-3alpha,7alpha-dihydroxy-5beta-cholan-24-oic acid6-ethyl-3,7-dihydroxycholan-24-oic acid6-alpha-ethylchenodeoxycholic acidCholan-24-oic acid, 6-ethyl-3,7-dihydroxy-, (3alpha,5beta,6alpha,7alpha)-(3alpha,5beta,6alpha,7alpha)-6-Ethyl-3,7-dihydroxycholan-24-oic acid(4R)-4-[(1R,3aS,3bS,4R,5R,5aS,7R,9aS,9bS,11aR)-5-ethyl-4,7-dihydroxy-9a,11a-dimethyl-hexadecahydro-1H-cyclopenta[a]phenanthren-1-yl]pentanoic acidObeticholicAcidacidum obeticholicum(4R)-4-((1R,3aS,3bS,4R,5R,5aS,7R,9aS,9bS,11aR)-5-ethyl-4,7-dihydroxy-9a,11a-dimethyl-hexadecahydro-1H-cyclopenta(a)phenanthren-1-yl)pentanoic acid6-ethyl chenodeoxycholic acidObetichloic acid6alpha-Ethyl-chenodeoxycholic acid
External Identifiers
EC NUMBER: 810-245-2DSSTOX SUBSTANCE ID: DTXSID20196671CHEMBL ID: CHEMBL566315CHEBI ID: CHEBI:43602UNII: 0462Z4S4OZDRUGBANK ID: DB05990KEGG ID: C15636KEGG ID: D09360METABOLOMICS WORKBENCH ID: 149608NCI THESAURUS CODE: C80837WIKIDATA ID: Q15708271
Literature & Patent References
DOI 10.1016/j.bmc.2025.118124Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocks.DOI 10.1016/j.ejmech.2024.117082Design, synthesis, and biological evaluation of novel highly potent FXR agonists bearing piperidine scaffold.DOI 10.1021/acs.jmedchem.4c01698Discovery of ZG-2305, an Orally Bioavailable Factor Inhibiting HIF Inhibitor for the Treatment of Obesity and Fatty Liver Disease.DOI 10.1021/acs.jmedchem.4c02720Discovery of First-in-Class FXR and HSD17B13 Dual Modulator for the Treatment of Metabolic Dysfunction-Associated Fatty Liver Disease.DOI 10.1021/acs.jmedchem.4c02809A Collection of Novel Antitumor Agents That Regulate Lipid Metabolism in the Tumor Microenvironment.DOI 10.1021/acs.jmedchem.5c00119Discovery of Highly Potent, Selective, and Liver-Targeting HSD17B13 Inhibitor with Robust In Vivo Anti-MASH Activity.DOI 10.1021/acs.jmedchem.5c00539Dual Modulator of FXR and HSD17B13: Revitalizing FXR Therapies in MASH.PMID 39432709Discovery of ZG-2305, an Orally Bioavailable Factor Inhibiting HIF Inhibitor for the Treatment of Obesity and Fatty Liver Disease.

Documentation & Compliance Facts

Compliance Facts

Shipment review: Required

Documentation available by request

Certificate of Analysis (COA): By request

Supplier Safety Data Sheet (SDS): By request

Purity and pack size confirmation: By request

Availability and lead time review: Confirmed by RFQ

Shipment documentation review: By request

For supplier-issued documentation by request, use the RFQ actions on this page.Review preliminary safety reference

What happens after RFQ

  1. 1We review the CAS identity, quantity, and documentation request.
  2. 2We check sourcing options, supplier availability, COA/SDS, purity, pack size, and lead time.
  3. 3We review destination and shipment documentation needs when applicable.
  4. 4We follow up with a quotation or clarification request.

Text Reference Cues

Show non-linked catalog cues

Non-public related references

benzyl (4R)-4-[(3R,5R,8S,9S,10R,13R,14S,17R)-6-ethylidene-3-hydroxy-10,13-dimethyl-7-oxo-2,3,4,5,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]pentanoateCAS 1352328-66-5

Non-public references are shown as text only and do not imply equivalence, availability, or shared use.

Catalog navigation

Related Catalog Entries

Other public CAS pages in this catalog. These links support navigation across additional intermediates and do not imply equivalence, availability, or shared use.

CAS 1352328-66-5benzyl (4R)-4-[(3R,5R,8S,9S,10R,13R,14S,17R)-6-ethylidene-3-hydroxy-10,13-dimethyl-7-oxo-2,3,4,5,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]pentanoateCAS 134678-17-4LamivudineCAS 181695-72-7ValdecoxibCAS 21829-25-4NifedipineCAS 128-13-2Ursodeoxycholic AcidCAS 265129-71-3GW-7647CAS 1002310-00-0Tert-butyl 1-(2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)ethylcarbamateCAS 1005174-17-3(E)-3-(2-Propyl-6-(trifluoromethyl)pyridin-3-yl)acrylic acidCAS 1018125-49-92-(3-Cyclopropyl-6-ethyl-4-(trifluoromethyl)-1H-pyrazolo[3,4-b]pyridin-1-yl)acetic acidCAS 1018128-07-8Isopropyl 4-chloro-2-methylquinoline-6-carboxylate

RFQ questions for CAS 459789-99-2

What are the key identifiers for Obeticholic Acid (CAS 459789-99-2)?

Obeticholic Acid is identified by CAS 459789-99-2, with molecular formula C26H44O4, molecular weight 420.6, InChIKey ZXERDUOLZKYMJM-ZWECCWDJSA-N.

Does CAS 459789-99-2 have reported biological target evidence?

ChEMBL contains qualifying experimental assay evidence associated with Bile acid receptor, G-protein coupled bile acid receptor 1, G-protein coupled bile acid receptor 1, Alpha-1A adrenergic receptor, Alpha-2A adrenergic receptor. These records do not establish therapeutic efficacy or clinical use.

Can I request a COA for CAS 459789-99-2?

Yes. Submit an RFQ and specify COA requirements. Lot-specific COA depends on supplier confirmation.

Can I request supplier SDS for Obeticholic Acid?

Yes. Supplier SDS can be requested through the RFQ workflow before handling, storage, shipment, or procurement decisions.

Is CAS 459789-99-2 available for quotation?

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